Construction of the Azacyclic Core of Tabernaemontanine-Related Alkaloids via Tandem Reformatsky Aza-Claisen Rearrangement

  • Suh, Young-Ger
  • Lim, Changjin
  • Sim, Jaehoon
  • Lee, Jae Kyun
  • Surh, Young-Joon
  • ... Paek, Seung-Mann
Citations

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9
Citations

SCOPUS

9

초록

A divergent synthetic methodology for a tabernaemontanine-related alkaloid was developed. The synthetic route features practical improvements in the Pictet-Spengler cyclization for the tetrahydro-fi-carboline intermediate and an unprecedented tandem Reformatsky aza-Claisen rearrangement to create the core carbon skeleton and stereochemistries of tabernaemontanine-related alkaloids.

키워드

ENANTIOSPECIFIC TOTAL-SYNTHESISINDOLE ALKALOIDSBISINDOLE ALKALOIDSTABEMAEMONTANAVOBASINE
제목
Construction of the Azacyclic Core of Tabernaemontanine-Related Alkaloids via Tandem Reformatsky Aza-Claisen Rearrangement
저자
Suh, Young-GerLim, ChangjinSim, JaehoonLee, Jae KyunSurh, Young-JoonPaek, Seung-Mann
DOI
10.1021/acs.joc.6b02648
발행일
2017-02-03
유형
Article
저널명
Journal of Organic Chemistry
82
3
페이지
1464 ~ 1470